Lidocaine Cream (5.0% w/w)
Healthy Inc is a specialized global supplier and exporter of advanced anesthetics, dermatology, and targeted topical therapeutics. We provide ultra-high-purity, kinetically optimized Lidocaine Cream, manufactured in WHO–GMP certified, high-precision specialized topical facilities. This “Amino-Amide Local Anesthetic” is a strategic export to cosmetic clinics, dermatology centers, and retail pharmacies, serving as the globally preferred intervention for surface anesthesia before minor skin procedures.
Product Overview
This formulation operates as a “Reversible Nerve Block.” It physically stops the initiation and conduction of nerve impulses by interfering with the exchange of ions across the nerve membrane.
Mechanism 1 (Sodium Channel Blockade): Lidocaine physically binds to the voltage-gated sodium channels on the neuronal membrane. This prevents the influx of sodium ions required for the nerve to “fire” a pain signal to the brain.
Mechanism 2 (High-Dermal Penetration): Unlike gels, the 5% cream utilizes a specialized emulsion base that physically drives the active ingredient through the Stratum Corneum (the outer skin barrier) to reach the deeper nerve endings in the dermis.
Mechanism 3 (Stabilized Membrane): By stabilizing the neuronal membrane, the cream ensures that even high-intensity stimuli (like a needle prick or laser pulse) do not trigger a pain response.
Product Composition & Strength
We supply this product in a Smooth, Non-Greasy Oil-in-Water Emulsion, optimized for rapid absorption and ease of removal before a procedure.
| Active Ingredient | Strength (w/w) | Primary Clinical Function |
| Lidocaine USP/BP | 5.0% | The Clinical Powerhouse: The highest OTC/Rx strength for deep skin numbing. |
| Excipients | Benzyl Alcohol / Cetyl Alcohol | The Flux Matrix: Engineered to maximize drug delivery while maintaining skin hydration. |
Technical & Logistics Specifications
HS Code: 3004.90.99 (Medicaments acting on the nervous system – Local Anesthetics)
CAS Number: 137-58-6 (Lidocaine)
Dosage Form: Topical Cream (O/W Emulsion)
Packaging: Laminated Aluminum or Plastic Tubes (15g / 20g / 30g / 50g). Our high-barrier packaging ensures 24-month stability in Zone IVb tropical climates.
Manufacturing Authority & Compliance
Emulsion Homogeneity: Our manufacturing process utilizes High-Shear Vacuum Homogenizers to ensure the Lidocaine is perfectly micronized and dispersed. This prevents “hot spots” of high concentration and ensures a consistent numbing effect across the entire treated area.
pH Optimization: We utilize Automated pH Buffering to ensure the cream is slightly alkaline. This physically increases the “un-ionized” form of Lidocaine, which is the form that most easily penetrates the skin barrier.
Primary Indications
Aesthetic Medicine: Numbing before Laser Hair Removal, Microneedling, and Dermal Fillers.
Dermatology: Pain relief for minor skin biopsies, wart removal, and molluscum treatment.
General Practice: Pre-treatment for Vaccinations and venipuncture (blood draws) in pediatric patients.
Aesthetics: Surface anesthesia for tattoo application and permanent makeup.
Dosage & Administration
Standard Regimen: Apply a thick layer (approx. 1g-2g per 10cm²) to the target area 30 to 60 minutes before the procedure.
Occlusion Tip: Covering the cream with a plastic wrap (occlusive dressing) physically forces the medicine deeper into the skin and prevents evaporation, significantly enhancing the numbing effect.
Removal: Wipe off the excess cream thoroughly with a sterile gauze before starting the procedure.
Safety Warning: External Use Only. Do not apply to broken, infected, or inflamed skin. Systemic Toxicity: Avoid applying to very large surface areas (more than 2% of body surface) to prevent Lidocaine from entering the bloodstream, which can cause heart or CNS issues. Contraindication: Do not use in patients with a known allergy to “amide-type” local anesthetics.
Global Export & Contract Manufacturing
Healthy Inc is a premier Anesthesia and Dermatology Pharmaceutical Exporter in India. As a verified Medicine Supplier in Mumbai, we offer flexible Third Party Manufacturing (Contract Manufacturing) for high-volume anesthetic creams. Whether you are an Aesthetic Clinic Chain in the Middle East or a B2B Pharma Marketplace partner in Africa or the CIS, we ensure secure, WHO-GMP compliant delivery.
Commercial Inquiries:
WhatsApp/Call: +91 7710003340
Email: info@healthyinc.co.in